PDB entry 1rhk
View 1rhk on RCSB PDB site
Description: Crystal structure of the complex of caspase-3 with a phenyl-propyl-ketone inhibitor
Class: hydrolase/hydrolase inhibitor
Keywords: cysteine protease, caspase-3, apopain, cpp32, yama, hydrolase-hydrolase inhibitor complex
Deposited on
2003-11-14, released
2004-05-11
The last revision prior to the SCOPe 2.08 freeze date was dated
2017-10-11, with a file datestamp of
2017-10-06.
Experiment type: XRAY
Resolution: 2.5 Å
R-factor: N/A
AEROSPACI score: 0.21
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Caspase-3
Species: Homo sapiens [TaxId:9606]
Gene: CASP3, CPP32
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d1rhk.1 - Chain 'B':
Compound: Caspase-3
Species: Homo sapiens [TaxId:9606]
Gene: CASP3, CPP32
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d1rhk.1 - Chain 'C':
Compound: acetyl-asp-glu-val-fpr
Species: synthetic, synthetic
Database cross-references and differences (RAF-indexed):
- Heterogens: HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>1rhkA (A:)
sgisldnsykmdypemglciiinnknfhkstgmtsrsgtdvdaanlretfrnlkyevrnk
ndltreeivelmrdvskedhskrssfvcvllshgeegiifgtngpvdlkkitnffrgdrc
rsltgkpklfiiqacrgteldcgietd
Sequence, based on observed residues (ATOM records): (download)
>1rhkA (A:)
dnsykmdypemglciiinnknfhkstgmtsrsgtdvdaanlretfrnlkyevrnkndltr
eeivelmrdvskedhskrssfvcvllshgeegiifgtngpvdlkkitnffrgdrcrsltg
kpklfiiqacrgteldcgie
- Chain 'B':
Sequence, based on SEQRES records: (download)
>1rhkB (B:)
sgvdddmachkipveadflyaystapgyyswrnskdgswfiqslcamlkqyadklefmhi
ltrvnrkvatefesfsfdatfhakkqipcivsmltkelyfyh
Sequence, based on observed residues (ATOM records): (download)
>1rhkB (B:)
kipveadflyaystapgyyswrnskdgswfiqslcamlkqyadklefmhiltrvnrkvat
efesfsfdatfhakkqipcivsmltkelyfy
- Chain 'C':
No sequence available.