PDB entry 1rgz

View 1rgz on RCSB PDB site
Description: Enterobacter cloacae GC1 Class C beta-Lactamase Complexed with Transition-State Analog of Cefotaxime
Class: hydrolase
Keywords: hydrolase, cephalosporinase, enzyme inhibition, phosphonate, beta-lactam antibiotics, drug design
Deposited on 2003-11-13, released 2004-04-06
The last revision prior to the SCOPe 2.05 freeze date was dated 2011-07-13, with a file datestamp of 2011-05-25.
Experiment type: XRAY
Resolution: 1.37 Å
R-factor: 0.142
AEROSPACI score: 0.74 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: class C beta-lactamase
    Species: Enterobacter cloacae [TaxId:550]
    Gene: bla
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.05: d1rgza_
  • Heterogens: PTX, GOL, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence; same for both SEQRES and ATOM records: (download)
    >1rgzA (A:)
    pvsekqlaevvantvtplmkaqsvpgmavaviyqgkphyytfgkadiaankpvtpqtlfe
    lgsisktftgvlggdaiargeislddpvtrywpqltgkqwqgirmldlatytagglplqv
    pdevtdnasllrfyqnwqpqwkpgttrlyanasiglfgalavkpsgmpyeqamttrvlkp
    lkldhtwinvpkaeeahyawgyrdgkavravrvspgmldaqaygvktnvqdmanwvmanm
    apenvadaslkqgialaqsrywrigsmyqglgwemlnwpveantvvegsdskvalaplpv
    aevnppappvkaswvhktgstggfgsyvafipekqigivmlantsypnparveaayhile
    alq