PDB entry 1r64
View 1r64 on RCSB PDB site
Description: The 2.2 A crystal structure of Kex2 protease in complex with Ac-Arg-Glu-Lys-boroArg peptidyl boronic acid inhibitor
Class: hydrolase/hydrolase inhibitor
Keywords: kex2, kexin, protease, protein convertase, prohormone processing, proprotein convertase, subtilisin, hydrolase-hydrolase inhibitor complex
Deposited on
2003-10-14, released
2004-03-09
The last revision prior to the SCOPe 2.03 freeze date was dated
2011-11-16, with a file datestamp of
2011-11-11.
Experiment type: XRAY
Resolution: 2.2 Å
R-factor: 0.197
AEROSPACI score: 0.4
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Kexin
Species: Saccharomyces cerevisiae [TaxId:4932]
Gene: KEX2 OR QDS1 OR YNL238W OR N1122
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.03: d1r64a1, d1r64a2 - Chain 'B':
Compound: Kexin
Species: Saccharomyces cerevisiae [TaxId:4932]
Gene: KEX2 OR QDS1 OR YNL238W OR N1122
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.03: d1r64b1, d1r64b2 - Chain 'C':
Compound: Ac-Arg-Glu-Lys-boroArg peptide inhibitor
Species: synthetic, synthetic
Database cross-references and differences (RAF-indexed):
- Chain 'D':
Compound: Ac-Arg-Glu-Lys-boroArg peptide inhibitor
Species: synthetic, synthetic
Database cross-references and differences (RAF-indexed):
- Heterogens: NAG, CA, K, BTB, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence; same for both SEQRES and ATOM records: (download)
>1r64A (A:)
llpvkeaedklsindplferqwhlvnpsfpgsdinvldlwynnitgagvvaaivddgldy
enedlkdnfcaegswdfndntnlpkprlsddyhgtrcageiaakkgnnfcgvgvgynaki
sgirilsgdittedeaasliygldvndiyscswgpaddgrhlqgpsdlvkkalvkgvteg
rdskgaiyvfasgnggtrgdncnydgytnsiysitigaidhkdlhppysegcsavmavty
ssgsgeyihssdingrcsnshggtsaaaplaagvytllleanpnltwrdvqylsilsavg
leknadgdwrdsamgkkyshrygfgkidahkliemsktwenvnaqtwfylptlyvsqstn
steetlesvitisekslqdanfkriehvtvtvdidteirgtttvdlispagiisnlgvvr
prdvssegfkdwtfmsvahwgengvgdwkikvkttenghridfhswrlklfgesidsskt
e
- Chain 'B':
Sequence; same for both SEQRES and ATOM records: (download)
>1r64B (B:)
llpvkeaedklsindplferqwhlvnpsfpgsdinvldlwynnitgagvvaaivddgldy
enedlkdnfcaegswdfndntnlpkprlsddyhgtrcageiaakkgnnfcgvgvgynaki
sgirilsgdittedeaasliygldvndiyscswgpaddgrhlqgpsdlvkkalvkgvteg
rdskgaiyvfasgnggtrgdncnydgytnsiysitigaidhkdlhppysegcsavmavty
ssgsgeyihssdingrcsnshggtsaaaplaagvytllleanpnltwrdvqylsilsavg
leknadgdwrdsamgkkyshrygfgkidahkliemsktwenvnaqtwfylptlyvsqstn
steetlesvitisekslqdanfkriehvtvtvdidteirgtttvdlispagiisnlgvvr
prdvssegfkdwtfmsvahwgengvgdwkikvkttenghridfhswrlklfgesidsskt
e
- Chain 'C':
No sequence available.
- Chain 'D':
No sequence available.