PDB entry 1q8u
View 1q8u on RCSB PDB site
Description: The Catalytic Subunit of cAMP-dependent Protein Kinase in Complex with Rho-kinase Inhibitor H-1152P
Class: Transferase/Transferase Inhibitor
Keywords: KINASE-INHIBITOR-COMPLEX, PHOSPHOTRANSFERASE/INHIBITOR, CAMP, PHOSPHORYLATION, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING, PKA, RHO-KINASE, Transferase/Transferase Inhibitor COMPLEX
Deposited on
2003-08-22, released
2003-12-16
The last revision prior to the SCOPe 2.01 freeze date was dated
2009-02-24, with a file datestamp of
2009-03-01.
Experiment type: XRAY
Resolution: 1.9 Å
R-factor: 0.173
AEROSPACI score: 0.5
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: cAMP-dependent protein kinase, alpha-catalytic subunit
Species: Bos taurus [TaxId:9913]
Gene: PRKACA
Database cross-references and differences (RAF-indexed):
- Uniprot P00517 (Start-349)
- modified residue (9)
- modified residue (196)
- modified residue (337)
Domains in SCOPe 2.01: d1q8ua_ - Chain 'B':
Compound: cAMP-dependent protein kinase inhibitor, alpha form
Species: synthetic, synthetic
Database cross-references and differences (RAF-indexed):
- Heterogens: H52, MG8, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>1q8uA (A:)
gnaaaakkgseqesvkeflakakedflkkwenpaqntahldqferiktlgtgsfgrvmlv
khmetgnhyamkildkqkvvklkqiehtlnekrilqavnfpflvklefsfkdnsnlymvm
eyvpggemfshlrrigrfsepharfyaaqivltfeylhsldliyrdlkpenllidqqgyi
qvtdfgfakrvkgrtwtlcgtpeylapeiilskgynkavdwwalgvliyemaagyppffa
dqpiqiyekivsgkvrfpshfssdlkdllrnllqvdltkrfgnlkngvndiknhkwfatt
dwiaiyqrkveapfipkfkgpgdtsnfddyeeeeirvsinekcgkefsef
Sequence, based on observed residues (ATOM records): (download)
>1q8uA (A:)
kkgseqesvkeflakakedflkkwenpaqntahldqferiktlgtgsfgrvmlvkhmetg
nhyamkildkqkvvklkqiehtlnekrilqavnfpflvklefsfkdnsnlymvmeyvpgg
emfshlrrigrfsepharfyaaqivltfeylhsldliyrdlkpenllidqqgyiqvtdfg
fakrvkgrtwtlcgtpeylapeiilskgynkavdwwalgvliyemaagyppffadqpiqi
yekivsgkvrfpshfssdlkdllrnllqvdltkrfgnlkngvndiknhkwfattdwiaiy
qrkveapfipkfkgpgdtsnfddyeeeeirvsinekcgkefsef
- Chain 'B':
No sequence available.