PDB entry 1pme
View 1pme on RCSB PDB site
Description: structure of penta mutant human erk2 map kinase complexed with a specific inhibitor of human p38 map kinase
Class: transferase
Keywords: map kinase, serine/threonine protein kinase, transferase
Deposited on
1998-06-08, released
1999-06-08
The last revision prior to the SCOPe 2.06 freeze date was dated
2009-02-24, with a file datestamp of
2009-03-01.
Experiment type: XRAY
Resolution: 2 Å
R-factor: 0.212
AEROSPACI score: 0.41
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: erk2
Species: Homo sapiens [TaxId:9606]
Gene: ERK2
Database cross-references and differences (RAF-indexed):
- Uniprot P28482 (Start-379)
- engineered (122)
- engineered (124-125)
- engineered (128-129)
- modified (180)
Domains in SCOPe 2.06: d1pmea_ - Heterogens: SO4, SB2, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>1pmeA (A:)
mssshhhhhhssglvprgshmaaaaaagagpemvrgqvfdvgprytnlsyigegaygmvc
saydnvnkvrvaikkispfehqtycqrtlreikillrfrheniigindiiraptieqmkd
vylvthlmgadlykllktqhlsndhicyflyqilrglkyihsanvlhrdlkpsnlllntt
cdlkicdfglarvadpdhdhtgflteyvatrwyrapeimlnskgytksidiwsvgcilae
mlsnrpifpgkhyldqlnhilgilgspsqedlnciinlkarnyllslphknkvpwnrlfp
nadskaldlldkmltfnphkrieveqalahpyleqyydpsdepiaeapfkfdmelddlpk
eklkelifeetarfqpgyrs
Sequence, based on observed residues (ATOM records): (download)
>1pmeA (A:)
gqvfdvgprytnlsyigygmvcsaydnvnkvrvaikkispfehqtycqrtlreikillrf
rheniigindiiraptieqmkdvylvthlmgadlykllktqhlsndhicyflyqilrglk
yihsanvlhrdlkpsnlllnttcdlkicdfglarvadpdhdhtgflteyvatrwyrapei
mlnskgytksidiwsvgcilaemlsnrpifpgkhyldqlnhilgilgspsqedlnciinl
karnyllslphknkvpwnrlfpnadskaldlldkmltfnphkrieveqalahpyleqyyd
psdepiaeapflpkeklkelifeetarfqpgyrs