PDB entry 1okz

View 1okz on RCSB PDB site
Description: structure of human pdk1 kinase domain in complex with ucn-01
Class: transferase
Keywords: protein kinase, pkb, pdk1, ucn-01, 7-hydroxy staurosporine, inhibitor, transferase, ATP-binding, phosphorylation
Deposited on 2003-08-01, released 2004-07-29
The last revision prior to the SCOP 1.73 freeze date was dated 2004-07-29, with a file datestamp of 2007-06-04.
Experiment type: XRAY
Resolution: 2.51 Å
R-factor: 0.19
AEROSPACI score: 0.34 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: 3-phosphoinositide dependent protein kinase 1
    Species: HOMO SAPIENS
    Database cross-references and differences (RAF-indexed): Domains in SCOP 1.73: d1okza_
  • Heterogens: SO4, UCN, GOL, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >1okzA (A:)
    mdgtaaeprpgagslqhaqpppqprkkrpedfkfgkilgegsfstvvlarelatsreyai
    kilekrhiikenkvpyvtrerdvmsrldhpffvklyftfqddeklyfglsyakngellky
    irkigsfdetctrfytaeivsaleylhgkgiihrdlkpenillnedmhiqitdfgtakvl
    speskqaransfvgtaqyvspellteksackssdlwalgciiyqlvaglppfragneyli
    fqkiikleydfpekffpkardlvekllvldatkrlgceemegygplkahpffesvtwenl
    hqqtppklta
    

    Sequence, based on observed residues (ATOM records): (download)
    >1okzA (A:)
    qprkkrpedfkfgkilgegsfstvvlarelatsreyaikilekrhiikenkvpyvtrerd
    vmsrldhpffvklyftfqddeklyfglsyakngellkyirkigsfdetctrfytaeivsa
    leylhgkgiihrdlkpenillnedmhiqitdfgtakvlnsfvgtaqyvspellteksack
    ssdlwalgciiyqlvaglppfragneylifqkiikleydfpekffpkardlvekllvlda
    tkrlgceemegygplkahpffesvtwenlhqqtppklt