PDB entry 1okz
View 1okz on RCSB PDB site
Description: structure of human pdk1 kinase domain in complex with ucn-01
Class: transferase
Keywords: protein kinase, pkb, pdk1, ucn-01, 7-hydroxy staurosporine, inhibitor, transferase, ATP-binding, phosphorylation
Deposited on
2003-08-01, released
2004-07-29
The last revision prior to the SCOP 1.73 freeze date was dated
2004-07-29, with a file datestamp of
2007-06-04.
Experiment type: XRAY
Resolution: 2.51 Å
R-factor: 0.19
AEROSPACI score: 0.34
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: 3-phosphoinositide dependent protein kinase 1
Species: HOMO SAPIENS
Database cross-references and differences (RAF-indexed):
Domains in SCOP 1.73: d1okza_ - Heterogens: SO4, UCN, GOL, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>1okzA (A:)
mdgtaaeprpgagslqhaqpppqprkkrpedfkfgkilgegsfstvvlarelatsreyai
kilekrhiikenkvpyvtrerdvmsrldhpffvklyftfqddeklyfglsyakngellky
irkigsfdetctrfytaeivsaleylhgkgiihrdlkpenillnedmhiqitdfgtakvl
speskqaransfvgtaqyvspellteksackssdlwalgciiyqlvaglppfragneyli
fqkiikleydfpekffpkardlvekllvldatkrlgceemegygplkahpffesvtwenl
hqqtppklta
Sequence, based on observed residues (ATOM records): (download)
>1okzA (A:)
qprkkrpedfkfgkilgegsfstvvlarelatsreyaikilekrhiikenkvpyvtrerd
vmsrldhpffvklyftfqddeklyfglsyakngellkyirkigsfdetctrfytaeivsa
leylhgkgiihrdlkpenillnedmhiqitdfgtakvlnsfvgtaqyvspellteksack
ssdlwalgciiyqlvaglppfragneylifqkiikleydfpekffpkardlvekllvlda
tkrlgceemegygplkahpffesvtwenlhqqtppklt