PDB entry 1nrl
View 1nrl on RCSB PDB site
Description: Crystal Structure of the human PXR-LBD in complex with an SRC-1 coactivator peptide and SR12813
Class: transcription
Keywords: nuclear receptor, coactivator, PXR, xenobiotic, SRC-1, ligand binding domain, TRANSCRIPTION
Deposited on
2003-01-25, released
2003-08-19
The last revision prior to the SCOPe 2.02 freeze date was dated
2009-02-24, with a file datestamp of
2009-03-01.
Experiment type: XRAY
Resolution: 2 Å
R-factor: 0.216
AEROSPACI score: 0.41
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: orphan nuclear receptor pxr
Species: Homo sapiens [TaxId:9606]
Gene: NR112 or PXR
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.02: d1nrla_ - Chain 'B':
Compound: orphan nuclear receptor pxr
Species: Homo sapiens [TaxId:9606]
Gene: NR112 or PXR
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.02: d1nrlb_ - Chain 'C':
Compound: Nuclear Receptor Coactivator 1 isoform 3
Species: synthetic, synthetic
Database cross-references and differences (RAF-indexed):
- Chain 'D':
Compound: Nuclear Receptor Coactivator 1 isoform 3
Species: synthetic, synthetic
Database cross-references and differences (RAF-indexed):
- Heterogens: SRL, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>1nrlA (A:)
mkkghhhhhhgsertgtqplgvqglteeqrmmirelmdaqmktfdttfshfknfrlpgvl
ssgcelpeslqapsreeaakwsqvrkdlcslkvslqlrgedgsvwnykppadsggkeifs
llphmadmstymfkgiisfakvisyfrdlpiedqisllkgaafelcqlrfntvfnaetgt
wecgrlsycledtaggfqqlllepmlkfhymlkklqlheeeyvlmqaislfspdrpgvlq
hrvvdqlqeqfaitlksyiecnrpqpahrflflkimamltelrsinaqhtqrllriqdih
pfatplmqelfgitgs
Sequence, based on observed residues (ATOM records): (download)
>1nrlA (A:)
glteeqrmmirelmdaqmktfdttfshfknfrlpgvsreeaakwsqvrkdlcslkvslql
rgedgsvwnykppadsggkeifsllphmadmstymfkgiisfakvisyfrdlpiedqisl
lkgaafelcqlrfntvfnaetgtwecgrlsycledtaggfqqlllepmlkfhymlkklql
heeeyvlmqaislfspdrpgvlqhrvvdqlqeqfaitlksyiecnrpqpahrflflkima
mltelrsinaqhtqrllriqdihpfatplmqelfgitg
- Chain 'B':
Sequence, based on SEQRES records: (download)
>1nrlB (B:)
mkkghhhhhhgsertgtqplgvqglteeqrmmirelmdaqmktfdttfshfknfrlpgvl
ssgcelpeslqapsreeaakwsqvrkdlcslkvslqlrgedgsvwnykppadsggkeifs
llphmadmstymfkgiisfakvisyfrdlpiedqisllkgaafelcqlrfntvfnaetgt
wecgrlsycledtaggfqqlllepmlkfhymlkklqlheeeyvlmqaislfspdrpgvlq
hrvvdqlqeqfaitlksyiecnrpqpahrflflkimamltelrsinaqhtqrllriqdih
pfatplmqelfgitgs
Sequence, based on observed residues (ATOM records): (download)
>1nrlB (B:)
glteeqrmmirelmdaqmktfdttfshfknfrlpgvreeaakwsqvrkdlcslkvslqlr
gedgsvwnykppadsggkeifsllphmadmstymfkgiisfakvisyfrdlpiedqisll
kgaafelcqlrfntvfnaetgtwecgrlsycledtaggfqqlllepmlkfhymlkklqlh
eeeyvlmqaislfspdrpgvlqhrvvdqlqeqfaitlksyiecnrpqpahrflflkimam
ltelrsinaqhtqrllriqdihpfatplmqelfgi
- Chain 'C':
No sequence available.
- Chain 'D':
No sequence available.