PDB entry 1mzn
View 1mzn on RCSB PDB site
Description: CRYSTAL STRUCTURE at 1.9 ANGSTROEMS RESOLUTION OF THE HOMODIMER OF HUMAN RXR ALPHA LIGAND BINDING DOMAIN BOUND TO THE SYNTHETIC AGONIST COMPOUND BMS 649 AND A COACTIVATOR PEPTIDE
Class: Transcription
Keywords: Transcription, Nuclear Receptor, Retinoic Acid Receptors, Agonist
Deposited on
2002-10-09, released
2002-10-23
The last revision prior to the SCOP 1.73 freeze date was dated
2002-10-23, with a file datestamp of
2007-06-04.
Experiment type: XRAY
Resolution: 1.9 Å
R-factor: 0.195
AEROSPACI score: 0.5
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: RXR retinoid X receptor
Species: HOMO SAPIENS
Database cross-references and differences (RAF-indexed):
Domains in SCOP 1.73: d1mzna_ - Chain 'B':
Compound: nuclear receptor coactivator 2
Species: synthetic, synthetic
Database cross-references and differences (RAF-indexed):
- Chain 'C':
Compound: RXR retinoid X receptor
Species: HOMO SAPIENS
Database cross-references and differences (RAF-indexed):
Domains in SCOP 1.73: d1mznc_ - Chain 'D':
Compound: nuclear receptor coactivator 2
Species: synthetic, synthetic
Database cross-references and differences (RAF-indexed):
- Chain 'E':
Compound: RXR retinoid X receptor
Species: HOMO SAPIENS
Database cross-references and differences (RAF-indexed):
Domains in SCOP 1.73: d1mzne_ - Chain 'F':
Compound: nuclear receptor coactivator 2
Species: synthetic, synthetic
Database cross-references and differences (RAF-indexed):
- Chain 'G':
Compound: RXR retinoid X receptor
Species: HOMO SAPIENS
Database cross-references and differences (RAF-indexed):
Domains in SCOP 1.73: d1mzng_ - Chain 'H':
Compound: nuclear receptor coactivator 2
Species: synthetic, synthetic
Database cross-references and differences (RAF-indexed):
- Heterogens: BM6, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>1mznA (A:)
tssanedmpverileaelavepktetyveanmglnpsspndpvtnicqaadkqlftlvew
akriphfselplddqvillragwnelliasfshrsiavkdgillatglhvhrnsahsagv
gaifdrvltelvskmrdmqmdktelgclraivlfnpdskglsnpaevealrekvyaslea
yckhkypeqpgrfaklllrlpalrsiglkclehlfffkligdtpidtflmemleaphqmt
Sequence, based on observed residues (ATOM records): (download)
>1mznA (A:)
nedmpverileaelavepktetyveanndpvtnicqaadkqlftlvewakriphfselpl
ddqvillragwnelliasfshrsiavkdgillatglhvhrnsahsagvgaifdrvltelv
skmrdmqmdktelgclraivlfnpdskglsnpaevealrekvyasleayckhkypeqpgr
faklllrlpalrsiglkclehlfffkligdtpidtflmemleap
- Chain 'B':
No sequence available.
- Chain 'C':
Sequence, based on SEQRES records: (download)
>1mznC (C:)
tssanedmpverileaelavepktetyveanmglnpsspndpvtnicqaadkqlftlvew
akriphfselplddqvillragwnelliasfshrsiavkdgillatglhvhrnsahsagv
gaifdrvltelvskmrdmqmdktelgclraivlfnpdskglsnpaevealrekvyaslea
yckhkypeqpgrfaklllrlpalrsiglkclehlfffkligdtpidtflmemleaphqmt
Sequence, based on observed residues (ATOM records): (download)
>1mznC (C:)
dmpverileaelavepdpvtnicqaadkqlftlvewakriphfselplddqvillragwn
elliasfshrsiavkdgillatglhvhrnsahsagvgaifdrvltelvskmrdmqmdkte
lgclraivlfnpdskglsnpaevealrekvyasleayckhkypeqpgrfaklllrlpalr
siglkclehlfffkligdtpidtflmemleap
- Chain 'D':
No sequence available.
- Chain 'E':
Sequence, based on SEQRES records: (download)
>1mznE (E:)
tssanedmpverileaelavepktetyveanmglnpsspndpvtnicqaadkqlftlvew
akriphfselplddqvillragwnelliasfshrsiavkdgillatglhvhrnsahsagv
gaifdrvltelvskmrdmqmdktelgclraivlfnpdskglsnpaevealrekvyaslea
yckhkypeqpgrfaklllrlpalrsiglkclehlfffkligdtpidtflmemleaphqmt
Sequence, based on observed residues (ATOM records): (download)
>1mznE (E:)
nedmpverileaelavepktetyveanndpvtnicqaadkqlftlvewakriphfselpl
ddqvillragwnelliasfshrsiavkdgillatglhvhrnsahsagvgaifdrvltelv
skmrdmqmdktelgclraivlfnpdskglsnpaevealrekvyasleayckhkypeqpgr
faklllrlpalrsiglkclehlfffkligdtpidtflmemleap
- Chain 'F':
No sequence available.
- Chain 'G':
Sequence, based on SEQRES records: (download)
>1mznG (G:)
tssanedmpverileaelavepktetyveanmglnpsspndpvtnicqaadkqlftlvew
akriphfselplddqvillragwnelliasfshrsiavkdgillatglhvhrnsahsagv
gaifdrvltelvskmrdmqmdktelgclraivlfnpdskglsnpaevealrekvyaslea
yckhkypeqpgrfaklllrlpalrsiglkclehlfffkligdtpidtflmemleaphqmt
Sequence, based on observed residues (ATOM records): (download)
>1mznG (G:)
dmpverileaelavepdpvtnicqaadkqlftlvewakriphfselplddqvillragwn
elliasfshrsiavkdgillatglhvhrnsahsagvgaifdrvltelvskmrdmqmdkte
lgclraivlfnpdskglsnpaevealrekvyasleayckhkypeqpgrfaklllrlpalr
siglkclehlfffkligdtpidtflmemleap
- Chain 'H':
No sequence available.