PDB entry 1k1t
View 1k1t on RCSB PDB site
Description: Combining Mutations in HIV-1 Protease to Understand Mechanisms of Resistance
Class: hydrolase/hydrolase inhibitor
Keywords: hiv-1 protease, mutant, dimer, inhibitor
Deposited on
2001-09-25, released
2002-07-10
The last revision prior to the SCOP 1.75 freeze date was dated
2003-04-01, with a file datestamp of
2007-06-04.
Experiment type: XRAY
Resolution: 1.2 Å
R-factor: 0.196
AEROSPACI score: 0.91
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: protease retropepsin
Species: Human immunodeficiency virus 1
Database cross-references and differences (RAF-indexed):
- Uniprot P04587
- engineered (6)
- engineered (32)
- engineered (44)
- engineered (62)
- engineered (66)
- engineered (81)
- engineered (94)
Domains in SCOP 1.75: d1k1ta_ - Chain 'B':
Compound: protease retropepsin
Species: Human immunodeficiency virus 1
Database cross-references and differences (RAF-indexed):
- Uniprot P04587 (0-98)
- engineered (6)
- engineered (32)
- engineered (44)
- engineered (62)
- engineered (66)
- engineered (81)
- engineered (94)
Domains in SCOP 1.75: d1k1tb_ - Chain 'C':
Compound: peptide inhibitor rv(dcl)fea(nle)
- Heterogens: SO4, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence; same for both SEQRES and ATOM records: (download)
>1k1tA (A:)
pqitlwkrplvtikiggqlkealldtgaddtvieemslpgrwkpimiggiggfikvrqyd
qiiieiaghkaigtvlvgptpsniigrnlltqigatlnf
- Chain 'B':
Sequence; same for both SEQRES and ATOM records: (download)
>1k1tB (B:)
pqitlwkrplvtikiggqlkealldtgaddtvieemslpgrwkpimiggiggfikvrqyd
qiiieiaghkaigtvlvgptpsniigrnlltqigatlnf
- Chain 'C':
No sequence available.