PDB entry 1jip

View 1jip on RCSB PDB site
Description: P450eryF(A245S)/ketoconazole
Class: hydrolase
Keywords: Cytochrome P450, P450eryF, P450eryF(A245S), ketoconazole, azole drug, HYDROLASE
Deposited on 2001-07-02, released 2001-10-17
The last revision prior to the SCOPe 2.03 freeze date was dated 2009-02-24, with a file datestamp of 2009-03-01.
Experiment type: XRAY
Resolution: 2 Å
R-factor: 0.21
AEROSPACI score: 0.43 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: cytochrome p450 107a1
    Species: Saccharopolyspora erythraea [TaxId:1836]
    Database cross-references and differences (RAF-indexed):
    • Uniprot Q00441 (0-402)
      • engineered (243)
    Domains in SCOPe 2.03: d1jipa_
  • Heterogens: HEM, KTN, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence; same for both SEQRES and ATOM records: (download)
    >1jipA (A:)
    ttvpdlesdsfhvdwyrtyaelretapvtpvrflgqdawlvtgydeakaalsdlrlssdp
    kkkypgvevefpaylgfpedvrnyfatnmgtsdppthtrlrklvsqeftvrrveamrprv
    eqitaelldevgdsgvvdivdrfahplpikvicellgvdekyrgefgrwsseilvmdper
    aeqrgqaarevvnfildlverrrtepgddllsalirvqddddgrlsadeltsialvllla
    gfessvsligigtylllthpdqlalvrrdpsalpnaveeilryiappetttrfaaeevei
    ggvaipqystvlvangaanrdpkqfpdphrfdvtrdtrghlsfgqgihfcmgrplakleg
    evalralfgrfpalslgidaddvvwrrslllrgidhlpvrldg