PDB entry 1c5o
View 1c5o on RCSB PDB site
Description: structural basis for selectivity of a small molecule, s1-binding, sub- micromolar inhibitor of urokinase type plasminogen activator
Deposited on
1999-12-22, released
2000-12-22
The last revision prior to the SCOP 1.57 freeze date was dated
2001-09-26, with a file datestamp of
2001-09-26.
Experiment type: XRAY
Resolution: 1.9 Å
R-factor: 0.2
AEROSPACI score: 0.45
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'H':
Domains in SCOP 1.57: d1c5o.1 - Chain 'L':
Domains in SCOP 1.57: d1c5o.1
PDB Chain Sequences:
- Chain 'H':
Sequence, based on SEQRES records: (download)
>1c5oH (H:)
ivegsdaeigmspwqvmlfrkspqellcgaslisdrwvltaahcllyppwdknftendll
vrigkhsrtryerniekismlekiyihprynwrenldrdialmklkkpvafsdyihpvcl
pdretaasllqagykgrvtgwgnlketwtanvgkgqpsvlqvvnlpiverpvckdstrir
itdnmfcagykpdegkrgdacegdsggpfvmkspfnnrwyqmgivswgegcdrdgkygfy
thvfrlkkwiqkvidqfge
Sequence, based on observed residues (ATOM records): (download)
>1c5oH (H:)
ivegsdaeigmspwqvmlfrkspqellcgaslisdrwvltaahcllyppwdknftendll
vrigkhsrtryerniekismlekiyihprynwrenldrdialmklkkpvafsdyihpvcl
pdretaasllqagykgrvtgwgnlketgqpsvlqvvnlpiverpvckdstriritdnmfc
agykpdegkrgdacegdsggpfvmkspfnnrwyqmgivswgegcdrdgkygfythvfrlk
kwiqkvidqfge
- Chain 'L':
Sequence; same for both SEQRES and ATOM records: (download)
>1c5oL (L:)
tfgsgeadcglrplfekksledkterellesyidgr