PDB entry 1c5l
View 1c5l on RCSB PDB site
Description: structural basis for selectivity of a small molecule, s1-binding, sub- micromolar inhibitor of urokinase type plasminogen activator
Deposited on
1999-12-22, released
2000-12-22
The last revision prior to the SCOP 1.71 freeze date was dated
2001-09-26, with a file datestamp of
2001-09-26.
Experiment type: XRAY
Resolution: 1.47 Å
R-factor: 0.215
AEROSPACI score: 0.58
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'H':
Domains in SCOP 1.71: d1c5l.1 - Chain 'L':
Domains in SCOP 1.71: d1c5l.1
PDB Chain Sequences:
- Chain 'H':
Sequence, based on SEQRES records: (download)
>1c5lH (H:)
ivegsdaeigmspwqvmlfrkspqellcgaslisdrwvltaahcllyppwdknftendll
vrigkhsrtryerniekismlekiyihprynwrenldrdialmklkkpvafsdyihpvcl
pdretaasllqagykgrvtgwgnlketwtanvgkgqpsvlqvvnlpiverpvckdstrir
itdnmfcagykpdegkrgdacegdsggpfvmkspfnnrwyqmgivswgegcdrdgkygfy
thvfrlkkwiqkvidqfge
Sequence, based on observed residues (ATOM records): (download)
>1c5lH (H:)
ivegsdaeigmspwqvmlfrkspqellcgaslisdrwvltaahcllyppwdknftendll
vrigkhsrtryerniekismlekiyihprynwrenldrdialmklkkpvafsdyihpvcl
pdretaasllqagykgrvtgwgnlketgqpsvlqvvnlpiverpvckdstriritdnmfc
agykpdegkrgdacegdsggpfvmkspfnnrwyqmgivswgegcdrdgkygfythvfrlk
kwiqkvidqfge
- Chain 'L':
Sequence; same for both SEQRES and ATOM records: (download)
>1c5lL (L:)
tfgsgeadcglrplfekksledkterellesyidgr